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Atomistry » Sodium » PDB 6sxg-6tbk » 6t8a | ||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Atomistry » Sodium » PDB 6sxg-6tbk » 6t8a » |
Sodium in PDB 6t8a: Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R)- 3-Cyclohexyl 2-((Phenylmethyl)Sulfonamido)Propanoyl)Pyrrolidine-2- Carboxamido)Methyl)Phosphonate (Mi-492)Enzymatic activity of Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R)- 3-Cyclohexyl 2-((Phenylmethyl)Sulfonamido)Propanoyl)Pyrrolidine-2- Carboxamido)Methyl)Phosphonate (Mi-492)
All present enzymatic activity of Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R)- 3-Cyclohexyl 2-((Phenylmethyl)Sulfonamido)Propanoyl)Pyrrolidine-2- Carboxamido)Methyl)Phosphonate (Mi-492):
3.4.21.5; Protein crystallography data
The structure of Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R)- 3-Cyclohexyl 2-((Phenylmethyl)Sulfonamido)Propanoyl)Pyrrolidine-2- Carboxamido)Methyl)Phosphonate (Mi-492), PDB code: 6t8a
was solved by
S.A.Ngaha,
A.Sandner,
S.Huber,
A.Heine,
T.Steinmetzer,
O.Pilgram,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Sodium Binding Sites:
The binding sites of Sodium atom in the Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R)- 3-Cyclohexyl 2-((Phenylmethyl)Sulfonamido)Propanoyl)Pyrrolidine-2- Carboxamido)Methyl)Phosphonate (Mi-492)
(pdb code 6t8a). This binding sites where shown within
5.0 Angstroms radius around Sodium atom.
In total 2 binding sites of Sodium where determined in the Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R)- 3-Cyclohexyl 2-((Phenylmethyl)Sulfonamido)Propanoyl)Pyrrolidine-2- Carboxamido)Methyl)Phosphonate (Mi-492), PDB code: 6t8a: Jump to Sodium binding site number: 1; 2; Sodium binding site 1 out of 2 in 6t8aGo back to Sodium Binding Sites List in 6t8a
Sodium binding site 1 out
of 2 in the Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R)- 3-Cyclohexyl 2-((Phenylmethyl)Sulfonamido)Propanoyl)Pyrrolidine-2- Carboxamido)Methyl)Phosphonate (Mi-492)
Mono view Stereo pair view
Sodium binding site 2 out of 2 in 6t8aGo back to Sodium Binding Sites List in 6t8a
Sodium binding site 2 out
of 2 in the Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R)- 3-Cyclohexyl 2-((Phenylmethyl)Sulfonamido)Propanoyl)Pyrrolidine-2- Carboxamido)Methyl)Phosphonate (Mi-492)
Mono view Stereo pair view
Reference:
S.A.Ngaha,
A.Sandner,
S.Huber,
O.Pilgram,
A.Heine,
T.Steinmetzer.
Thrombin in Complex with Diphenyl ((4-Carbamimidoylphenyl)((S)-1-((R) -3-Cyclohexyl-2-((Phenylmethyl)Sulfonamido)Propanoyl) Pyrrolidine-2-Carboxamido)Methyl)Phosphonate (Mi-492) To Be Published.
Page generated: Tue Dec 15 13:04:41 2020
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