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Atomistry » Sodium » PDB 1t4b-1u8r » 1tbz | ||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Atomistry » Sodium » PDB 1t4b-1u8r » 1tbz » |
Sodium in PDB 1tbz: Human Thrombin with Active Site N-Methyl-D Phenylalanyl-N-[5- (Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L- Prolinamide Trifluroacetate and Exosite-HirugenEnzymatic activity of Human Thrombin with Active Site N-Methyl-D Phenylalanyl-N-[5- (Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L- Prolinamide Trifluroacetate and Exosite-Hirugen
All present enzymatic activity of Human Thrombin with Active Site N-Methyl-D Phenylalanyl-N-[5- (Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L- Prolinamide Trifluroacetate and Exosite-Hirugen:
3.4.21.5; Protein crystallography data
The structure of Human Thrombin with Active Site N-Methyl-D Phenylalanyl-N-[5- (Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L- Prolinamide Trifluroacetate and Exosite-Hirugen, PDB code: 1tbz
was solved by
J.H.Matthews,
R.Krishnan,
M.J.Costanzo,
B.E.Maryanoff,
A.Tulinsky,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Sodium Binding Sites:
The binding sites of Sodium atom in the Human Thrombin with Active Site N-Methyl-D Phenylalanyl-N-[5- (Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L- Prolinamide Trifluroacetate and Exosite-Hirugen
(pdb code 1tbz). This binding sites where shown within
5.0 Angstroms radius around Sodium atom.
In total 2 binding sites of Sodium where determined in the Human Thrombin with Active Site N-Methyl-D Phenylalanyl-N-[5- (Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L- Prolinamide Trifluroacetate and Exosite-Hirugen, PDB code: 1tbz: Jump to Sodium binding site number: 1; 2; Sodium binding site 1 out of 2 in 1tbzGo back to![]() ![]()
Sodium binding site 1 out
of 2 in the Human Thrombin with Active Site N-Methyl-D Phenylalanyl-N-[5- (Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L- Prolinamide Trifluroacetate and Exosite-Hirugen
![]() Mono view ![]() Stereo pair view
Sodium binding site 2 out of 2 in 1tbzGo back to![]() ![]()
Sodium binding site 2 out
of 2 in the Human Thrombin with Active Site N-Methyl-D Phenylalanyl-N-[5- (Aminoiminomethyl)Amino]-1-{{Benzothiazolyl)Carbonyl] Butyl]-L- Prolinamide Trifluroacetate and Exosite-Hirugen
![]() Mono view ![]() Stereo pair view
Reference:
J.H.Matthews,
R.Krishnan,
M.J.Costanzo,
B.E.Maryanoff,
A.Tulinsky.
Crystal Structures of Thrombin with Thiazole-Containing Inhibitors: Probes of the S1' Binding Site. Biophys.J. V. 71 2830 1996.
Page generated: Sun Oct 6 22:38:30 2024
ISSN: ISSN 0006-3495 PubMed: 8913620 |
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