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Atomistry » Sodium » PDB 1det-1ev6 » 1eas » |
Sodium in PDB 1eas: Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin- 2-One Trifluoromethyl KetonesEnzymatic activity of Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin- 2-One Trifluoromethyl Ketones
All present enzymatic activity of Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin- 2-One Trifluoromethyl Ketones:
3.4.21.36; Protein crystallography data
The structure of Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin- 2-One Trifluoromethyl Ketones, PDB code: 1eas
was solved by
C.Ceccarelli,
with X-Ray Crystallography technique. A brief refinement statistics is given in the table below:
Other elements in 1eas:
The structure of Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin- 2-One Trifluoromethyl Ketones also contains other interesting chemical elements:
Sodium Binding Sites:
The binding sites of Sodium atom in the Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin- 2-One Trifluoromethyl Ketones
(pdb code 1eas). This binding sites where shown within
5.0 Angstroms radius around Sodium atom.
In total only one binding site of Sodium was determined in the Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin- 2-One Trifluoromethyl Ketones, PDB code: 1eas: Sodium binding site 1 out of 1 in 1easGo back to Sodium Binding Sites List in 1eas
Sodium binding site 1 out
of 1 in the Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin- 2-One Trifluoromethyl Ketones
Mono view Stereo pair view
Reference:
P.R.Bernstein,
D.Andisik,
P.K.Bradley,
C.B.Bryant,
C.Ceccarelli,
J.R.Damewood Jr.,
R.Earley,
P.D.Edwards,
S.Feeney,
B.C.Gomes,
B.J.Kosmider,
G.B.Steelman,
R.M.Thomas,
E.P.Vacek,
C.A.Veale,
J.C.Williams,
D.J.Wolanin,
J.A.Woolson.
Nonpeptidic Inhibitors of Human Leukocyte Elastase. 3. Design, Synthesis, X-Ray Crystallographic Analysis, and Structure-Activity Relationships For A Series of Orally Active 3-Amino-6-Phenylpyridin-2-One Trifluoromethyl Ketones. J.Med.Chem. V. 37 3313 1994.
Page generated: Tue Dec 15 05:23:26 2020
ISSN: ISSN 0022-2623 PubMed: 7932559 DOI: 10.1021/JM00046A016 |
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